CATH Classification

Domain Context

CATH Clusters

Superfamily Histidine kinase-like ATPase, C-terminal domain
Functional Family Heat shock protein HSP 90-alpha

Enzyme Information

UniProtKB Entries (1)

P07900
HS90A_HUMAN
Homo sapiens
Heat shock protein HSP 90-alpha

PDB Structure

PDB 3HHU
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Potent triazolothione inhibitor of heat-shock protein-90.
Feldman, R.I., Mintzer, B., Zhu, D., Wu, J.M., Biroc, S.L., Yuan, S., Emayan, K., Chang, Z., Chen, D., Arnaiz, D.O., Bryant, J., Ge, X.S., Whitlow, M., Adler, M., Polokoff, M.A., Li, W.W., Ferrer, M., Sato, T., Gu, J.M., Shen, J., Tseng, J.L., Dinter, H., Buckman, B.
Chem.Biol.Drug Des.