CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Peroxisome proliferator-activated receptor gamma

Enzyme Information

UniProtKB Entries (1)

P37231
PPARG_HUMAN
Homo sapiens
Peroxisome proliferator-activated receptor gamma

PDB Structure

PDB 3BC5
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Design, synthesis and structure-activity relationships of azole acids as novel, potent dual PPAR alpha/gamma agonists.
Zhang, H., Ryono, D.E., Devasthale, P., Wang, W., O'Malley, K., Farrelly, D., Gu, L., Harrity, T., Cap, M., Chu, C., Locke, K., Zhang, L., Lippy, J., Kunselman, L., Morgan, N., Flynn, N., Moore, L., Hosagrahara, V., Zhang, L., Kadiyala, P., Xu, C., Doweyko, A.M., Bell, A., Chang, C., Muckelbauer, J., Zahler, R., Hariharan, N., Cheng, P.T.
Bioorg.Med.Chem.Lett.