CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Androgen receptor variant

Enzyme Information

UniProtKB Entries (1)

P10275
ANDR_HUMAN
Homo sapiens
Androgen receptor

PDB Structure

PDB 2PNU
External Links
Method X-RAY DIFFRACTION
Organism Escherichia
Primary Citation
Structural Characterization of the Human Androgen Receptor Ligand-binding Domain Complexed with EM5744, a Rationally Designed Steroidal Ligand Bearing a Bulky Chain Directed toward Helix 12.
Cantin, L., Faucher, F., Couture, J.F., de Jesus-Tran, K.P., Legrand, P., Ciobanu, L.C., Frechette, Y., Labrecque, R., Singh, S.M., Labrie, F., Breton, R.
J.Biol.Chem.