CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Androgen receptor variant

Enzyme Information

UniProtKB Entries (1)

P15207
ANDR_RAT
Rattus norvegicus
Androgen receptor

PDB Structure

PDB 2IHQ
External Links
Method X-RAY DIFFRACTION
Organism Escherichia
Primary Citation
Discovery of potent, orally-active, and muscle-selective androgen receptor modulators based on an N-aryl-hydroxybicyclohydantoin scaffold.
Sun, C., Robl, J.A., Wang, T.C., Huang, Y., Kuhns, J.E., Lupisella, J.A., Beehler, B.C., Golla, R., Sleph, P.G., Seethala, R., Fura, A., Krystek, S.R., An, Y., Malley, M.F., Sack, J.S., Salvati, M.E., Grover, G.J., Ostrowski, J., Hamann, L.G.
J.Med.Chem.