CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Estrogen receptor

Enzyme Information

UniProtKB Entries (1)

P03372
ESR1_HUMAN
Homo sapiens
Estrogen receptor

PDB Structure

PDB 1XP9
External Links
Method X-RAY DIFFRACTION
Organism Escherichia
Primary Citation
Estrogen receptor ligands. Part 9: Dihydrobenzoxathiin SERAMs with alkyl substituted pyrrolidine side chains and linkers.
Blizzard, T.A., Dininno, F., Morgan, J.D., Chen, H.Y., Wu, J.Y., Kim, S., Chan, W., Birzin, E.T., Yang, Y.T., Pai, L.Y., Fitzgerald, P.M., Sharma, N., Li, Y., Zhang, Z., Hayes, E.C., Dasilva, C.A., Tang, W., Rohrer, S.P., Schaeffer, J.M., Hammond, M.L.
Bioorg.Med.Chem.Lett.