PDB Information

PDB6T3C
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
The discovery of 7-methyl-2-[(7-methyl[1,2,4]triazolo[1,5-a]pyridin-6-yl)amino]-9-(tetrahydro-2H-pyran-4-yl)-7,9-dihydro-8H-purin-8-one (AZD7648), a potent and selective DNA-dependent protein kinase (DNA-PK) inhibitor.
Goldberg, F.W., Finlay, M.R.V., Ting, A., Beattie, D., Lamont, G., Fallan, C., Wrigley, G., Schimpl, M., Howard, M.R., Williamson, B., Vazquez-Chantada, M., Barratt, D., Davies, B., Cadogan, E., Ramos Montoya, A., Dean, E.
J.Med.Chem.
HeaderTransferase
Released2019-10-10
Resolution2.620
CATH Insert Date05 Jan, 2020

PDB Images (1)

PDB Prints

PDB Chains (0)

Chain ID Date inserted into CATH CATH Status

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (0)

Accession Gene ID Taxon Description