PDB Information

PDB6T3B
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
The discovery of 7-methyl-2-[(7-methyl[1,2,4]triazolo[1,5-a]pyridin-6-yl)amino]-9-(tetrahydro-2H-pyran-4-yl)-7,9-dihydro-8H-purin-8-one (AZD7648), a potent and selective DNA-dependent protein kinase (DNA-PK) inhibitor.
Goldberg, F.W., Finlay, M.R.V., Ting, A., Beattie, D., Lamont, G., Fallan, C., Wrigley, G., Schimpl, M., Howard, M.R., Williamson, B., Vazquez-Chantada, M., Barratt, D., Davies, B., Cadogan, E., Ramos Montoya, A., Dean, E.
J.Med.Chem.
HeaderTransferase
Released2019-10-10
Resolution3.010
CATH Insert Date05 Jan, 2020

PDB Images (1)

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PDB Chains (0)

Chain ID Date inserted into CATH CATH Status

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (0)

Accession Gene ID Taxon Description