PDB Information

PDB6S57
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
A Qualified Success: Discovery of a New Series of ATAD2 Bromodomain Inhibitors with a Novel Binding Mode Using High-Throughput Screening and Hit Qualification.
Bamborough, P., Chung, C.W., Demont, E.H., Bridges, A.M., Craggs, P.D., Dixon, D.P., Francis, P., Furze, R.C., Grandi, P., Jones, E.J., Karamshi, B., Locke, K., Lucas, S.C.C., Michon, A.M., Mitchell, D.J., Pogany, P., Prinjha, R.K., Rau, C., Roa, A.M., Roberts, A.D., Sheppard, R.J., Watson, R.J.
J.Med.Chem.
HeaderTranscription
Released2019-06-30
Resolution1.820
CATH Insert Date01 Sep, 2019

PDB Images (2)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 01 Sep, 2019 New

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (0)

Accession Gene ID Taxon Description