PDB Information

PDB6QXU
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery and Optimization of 2-Arylquinazolin-4-ones into a Potent and Selective Tankyrase Inhibitor Modulating Wnt Pathway Activity.
Buchstaller, H.P., Anlauf, U., Dorsch, D., Kuhn, D., Lehmann, M., Leuthner, B., Musil, D., Radtki, D., Ritzert, C., Rohdich, F., Schneider, R., Esdar, C.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2019-03-08
Resolution1.200
CATH Insert Date18 Aug, 2019

PDB Images (2)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 18 Aug, 2019 New

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (0)

Accession Gene ID Taxon Description