PDB Information

PDB6OIN
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A.
Leaver, D.J., Cleary, B., Nguyen, N., Priebbenow, D.L., Lagiakos, H.R., Sanchez, J., Xue, L., Huang, F., Sun, Y., Mujumdar, P., Mudududdla, R., Varghese, S., Teguh, S., Charman, S.A., White, K.L., Katneni, K., Cuellar, M., Strasser, J.M., Dahlin, J.L., Walters, M.A., Street, I.P., Monahan, B.J., Jarman, K.E., Sabroux, H.J., Falk, H., Chung, M.C., Hermans, S.J., Parker, M.W., Thomas, T., Baell, J.B.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2019-04-09
Resolution1.700
CATH Insert Date07 Jul, 2019

PDB Images (2)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 07 Jul, 2019 New

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (0)

Accession Gene ID Taxon Description