PDB Information

PDB6O95
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Development of Potent and Selective Pyrazolopyrimidine IRAK4 Inhibitors.
Bryan, M.C., Drobnick, J., Gobbi, A., Kolesnikov, A., Chen, Y., Rajapaksa, N., Ndubaku, C., Feng, J., Chang, W., Francis, R., Yu, C., Choo, E.F., DeMent, K., Ran, Y., An, L., Emson, C., Huang, Z., Sujatha-Bhaskar, S., Brightbill, H., DiPasquale, A., Maher, J., Wai, J., McKenzie, B.S., Lupardus, P.J., Zarrin, A.A., Kiefer, J.R.
J.Med.Chem.
HeaderImmune System
Released2019-03-13
Resolution1.770
CATH Insert Date26 May, 2019

PDB Images (5)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 26 May, 2019 Holding pen
B 26 May, 2019 Holding pen
C 26 May, 2019 Holding pen
D 26 May, 2019 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q9NWZ3 IRAK4_HUMAN Homo sapiens Interleukin-1 receptor-associated kinase 4
Q9NWZ3 IRAK4_HUMAN Homo sapiens Interleukin-1 receptor-associated kinase 4
Q9NWZ3 IRAK4_HUMAN Homo sapiens Interleukin-1 receptor-associated kinase 4
Q9NWZ3 IRAK4_HUMAN Homo sapiens Interleukin-1 receptor-associated kinase 4