PDB Information

PDB6NPV
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera aff. frugiperda 2 RZ-2014
Gene SourceHomo sapiens
Primary Citation
Identification and Optimization of Novel Small c-Abl Kinase Activators Using Fragment and HTS Methodologies.
Simpson, G.L., Bertrand, S.M., Borthwick, J.A., Campobasso, N., Chabanet, J., Chen, S., Coggins, J., Cottom, J., Christensen, S.B., Dawson, H.C., Evans, H.L., Hobbs, A.N., Hong, X., Mangatt, B., Munoz-Muriedas, J., Oliff, A., Qin, D., Scott-Stevens, P., Ward, P., Washio, Y., Yang, J., Young, R.J.
J. Med. Chem.
HeaderTransferase
Released2019-01-18
Resolution1.860
CATH Insert Date17 Mar, 2019

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 17 Mar, 2019 Chopped
B 17 Mar, 2019 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
6npvA01 18 Mar, 2019 3.30.200.20 Assigned
6npvA02 18 Mar, 2019 1.10.510.10 Assigned
6npvB01 18 Mar, 2019 3.30.200.20 Assigned
6npvB02 18 Mar, 2019 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00519 ABL1_HUMAN Homo sapiens Tyrosine-protein kinase ABL1
P00519 ABL1_HUMAN Homo sapiens Tyrosine-protein kinase ABL1