PDB Information

PDB6J3P
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of Pyrrolo[3,2- d]pyrimidin-4-one Derivatives as a New Class of Potent and Cell-Active Inhibitors of P300/CBP-Associated Factor Bromodomain.
Huang, L., Li, H., Li, L., Niu, L., Seupel, R., Wu, C., Cheng, W., Chen, C., Ding, B., Brennan, P.E., Yang, S.
J.Med.Chem.
HeaderTransferase
Released2019-01-05
Resolution1.600
CATH Insert Date05 May, 2019

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 May, 2019 Chopped
B 05 May, 2019 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6j3pA00 06 May, 2019 1.20.920.10 Assigned
6j3pB00 06 May, 2019 1.20.920.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q92830 KAT2A_HUMAN Homo sapiens Histone acetyltransferase KAT2A
Q92830 KAT2A_HUMAN Homo sapiens Histone acetyltransferase KAT2A