PDB 6iji
PDB Information
| PDB | 6IJI |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21 |
| Gene Source | Homo sapiens |
| Primary Citation | Validation of Phosphodiesterase-10 as a Novel Target for Pulmonary Arterial Hypertension via Highly Selective and Subnanomolar Inhibitors.
J. Med. Chem.
|
| Header | Hydrolase/Inhibitor |
| Released | 2018-10-10 |
| Resolution | 2.700 |
| CATH Insert Date | 14 Apr, 2019 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 14 Apr, 2019 | Chopped |
| B | 14 Apr, 2019 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 6ijiA00 | 15 Apr, 2019 | 1.10.1300.10 | Assigned |
| 6ijiB00 | 15 Apr, 2019 | 1.10.1300.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q9Y233 | PDE10_HUMAN | Homo sapiens | cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A |
| Q9Y233 | PDE10_HUMAN | Homo sapiens | cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A |
