PDB Information

PDB6HTR
MethodX-RAY DIFFRACTION
Host OrganismSaccharomyces cerevisiae S288c
Gene SourceHomo sapiens
Primary Citation
Structure-Based Design of Inhibitors Selective for Human Proteasome beta 2c or beta 2i Subunits.
Xin, B.T., Huber, E.M., de Bruin, G., Heinemeyer, W., Maurits, E., Espinal, C., Du, Y., Janssens, M., Weyburne, E.S., Kisselev, A.F., Florea, B.I., Driessen, C., van der Marel, G.A., Groll, M., Overkleeft, H.S.
J.Med.Chem.
HeaderHydrolase
Released2018-10-04
Resolution2.600
CATH Insert Date03 Feb, 2019

PDB Images (57)

PDB Prints

PDB Chains (28)

Chain ID Date inserted into CATH CATH Status
a 03 Feb, 2019 Chopped
A 03 Feb, 2019 Chopped
b 03 Feb, 2019 Chopped
B 03 Feb, 2019 Chopped
C 03 Feb, 2019 Chopped
D 03 Feb, 2019 Chopped
E 03 Feb, 2019 Chopped
F 03 Feb, 2019 Chopped
G 03 Feb, 2019 Chopped
H 03 Feb, 2019 Chopped
I 03 Feb, 2019 Chopped
J 03 Feb, 2019 Chopped
K 03 Feb, 2019 Chopped
L 03 Feb, 2019 Chopped
M 03 Feb, 2019 Chopped
N 03 Feb, 2019 Chopped
O 03 Feb, 2019 Chopped
P 03 Feb, 2019 Chopped
Q 03 Feb, 2019 Chopped
R 03 Feb, 2019 Chopped
S 03 Feb, 2019 Chopped
T 03 Feb, 2019 Chopped
U 03 Feb, 2019 Chopped
V 03 Feb, 2019 Chopped
W 03 Feb, 2019 Chopped
X 03 Feb, 2019 Chopped
Y 03 Feb, 2019 Chopped
Z 03 Feb, 2019 Chopped

CATH Domains (28)

Domain ID Date inserted into CATH Superfamily CATH Status
6htra00 04 Feb, 2019 3.60.20.10 Assigned
6htrA00 04 Feb, 2019 3.60.20.10 Assigned
6htrb00 04 Feb, 2019 3.60.20.10 Assigned
6htrB00 04 Feb, 2019 3.60.20.10 Assigned
6htrC00 04 Feb, 2019 3.60.20.10 Assigned
6htrD00 04 Feb, 2019 3.60.20.10 Assigned
6htrE00 04 Feb, 2019 3.60.20.10 Assigned
6htrF00 04 Feb, 2019 3.60.20.10 Assigned
6htrG00 04 Feb, 2019 3.60.20.10 Assigned
6htrH00 04 Feb, 2019 3.60.20.10 Assigned
6htrI00 04 Feb, 2019 3.60.20.10 Assigned
6htrJ00 04 Feb, 2019 3.60.20.10 Assigned
6htrK00 04 Feb, 2019 3.60.20.10 Assigned
6htrL00 04 Feb, 2019 3.60.20.10 Assigned
6htrM00 04 Feb, 2019 3.60.20.10 Assigned
6htrN00 04 Feb, 2019 3.60.20.10 Assigned
6htrO00 04 Feb, 2019 3.60.20.10 Assigned
6htrP00 04 Feb, 2019 3.60.20.10 Assigned
6htrQ00 04 Feb, 2019 3.60.20.10 Assigned
6htrR00 04 Feb, 2019 3.60.20.10 Assigned
6htrS00 04 Feb, 2019 3.60.20.10 Assigned
6htrT00 04 Feb, 2019 3.60.20.10 Assigned
6htrU00 04 Feb, 2019 3.60.20.10 Assigned
6htrV00 04 Feb, 2019 3.60.20.10 Assigned
6htrW00 04 Feb, 2019 3.60.20.10 Assigned
6htrX00 04 Feb, 2019 3.60.20.10 Assigned
6htrY00 04 Feb, 2019 3.60.20.10 Assigned
6htrZ00 04 Feb, 2019 3.60.20.10 Assigned

UniProtKB Entries (28)

Accession Gene ID Taxon Description
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
Q99436 PSB7_HUMAN Homo sapiens Proteasome subunit beta type-7
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
Q99436 PSB7_HUMAN Homo sapiens Proteasome subunit beta type-7
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5