PDB Information

PDB6HTB
MethodX-RAY DIFFRACTION
Host OrganismSaccharomyces cerevisiae S288c
Gene SourceHomo sapiens
Primary Citation
Structure-Based Design of Inhibitors Selective for Human Proteasome beta 2c or beta 2i Subunits.
Xin, B.T., Huber, E.M., de Bruin, G., Heinemeyer, W., Maurits, E., Espinal, C., Du, Y., Janssens, M., Weyburne, E.S., Kisselev, A.F., Florea, B.I., Driessen, C., van der Marel, G.A., Groll, M., Overkleeft, H.S.
J.Med.Chem.
HeaderHydrolase
Released2018-10-03
Resolution2.700
CATH Insert Date03 Feb, 2019

PDB Images (57)

PDB Prints

PDB Chains (28)

Chain ID Date inserted into CATH CATH Status
a 03 Feb, 2019 Chopped
A 03 Feb, 2019 Chopped
b 03 Feb, 2019 Chopped
B 03 Feb, 2019 Chopped
C 03 Feb, 2019 Chopped
D 03 Feb, 2019 Chopped
E 03 Feb, 2019 Chopped
F 03 Feb, 2019 Chopped
G 03 Feb, 2019 Chopped
H 03 Feb, 2019 Chopped
I 03 Feb, 2019 Chopped
J 03 Feb, 2019 Chopped
K 03 Feb, 2019 Chopped
L 03 Feb, 2019 Chopped
M 03 Feb, 2019 Chopped
N 03 Feb, 2019 Chopped
O 03 Feb, 2019 Chopped
P 03 Feb, 2019 Chopped
Q 03 Feb, 2019 Chopped
R 03 Feb, 2019 Chopped
S 03 Feb, 2019 Chopped
T 03 Feb, 2019 Chopped
U 03 Feb, 2019 Chopped
V 03 Feb, 2019 Chopped
W 03 Feb, 2019 Chopped
X 03 Feb, 2019 Chopped
Y 03 Feb, 2019 Chopped
Z 03 Feb, 2019 Chopped

CATH Domains (28)

Domain ID Date inserted into CATH Superfamily CATH Status
6htba00 04 Feb, 2019 3.60.20.10 Assigned
6htbA00 04 Feb, 2019 3.60.20.10 Assigned
6htbb00 04 Feb, 2019 3.60.20.10 Assigned
6htbB00 04 Feb, 2019 3.60.20.10 Assigned
6htbC00 04 Feb, 2019 3.60.20.10 Assigned
6htbD00 04 Feb, 2019 3.60.20.10 Assigned
6htbE00 04 Feb, 2019 3.60.20.10 Assigned
6htbF00 04 Feb, 2019 3.60.20.10 Assigned
6htbG00 04 Feb, 2019 3.60.20.10 Assigned
6htbH00 04 Feb, 2019 3.60.20.10 Assigned
6htbI00 04 Feb, 2019 3.60.20.10 Assigned
6htbJ00 04 Feb, 2019 3.60.20.10 Assigned
6htbK00 04 Feb, 2019 3.60.20.10 Assigned
6htbL00 04 Feb, 2019 3.60.20.10 Assigned
6htbM00 04 Feb, 2019 3.60.20.10 Assigned
6htbN00 04 Feb, 2019 3.60.20.10 Assigned
6htbO00 04 Feb, 2019 3.60.20.10 Assigned
6htbP00 04 Feb, 2019 3.60.20.10 Assigned
6htbQ00 04 Feb, 2019 3.60.20.10 Assigned
6htbR00 04 Feb, 2019 3.60.20.10 Assigned
6htbS00 04 Feb, 2019 3.60.20.10 Assigned
6htbT00 04 Feb, 2019 3.60.20.10 Assigned
6htbU00 04 Feb, 2019 3.60.20.10 Assigned
6htbV00 04 Feb, 2019 3.60.20.10 Assigned
6htbW00 04 Feb, 2019 3.60.20.10 Assigned
6htbX00 04 Feb, 2019 3.60.20.10 Assigned
6htbY00 04 Feb, 2019 3.60.20.10 Assigned
6htbZ00 04 Feb, 2019 3.60.20.10 Assigned

UniProtKB Entries (28)

Accession Gene ID Taxon Description
Q99436 PSB7_HUMAN Homo sapiens Proteasome subunit beta type-7
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
Q99436 PSB7_HUMAN Homo sapiens Proteasome subunit beta type-7
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5