PDB Information

PDB6HSG
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceSchistosoma mansoni
Primary Citation
Characterization of Histone Deacetylase 8 (HDAC8) Selective Inhibition Reveals Specific Active Site Structural and Functional Determinants.
Marek, M., Shaik, T.B., Heimburg, T., Chakrabarti, A., Lancelot, J., Ramos-Morales, E., Da Veiga, C., Kalinin, D., Melesina, J., Robaa, D., Schmidtkunz, K., Suzuki, T., Holl, R., Ennifar, E., Pierce, R.J., Jung, M., Sippl, W., Romier, C.
J. Med. Chem.
HeaderHydrolase
Released2018-10-01
Resolution1.850
CATH Insert Date16 Dec, 2018

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 16 Dec, 2018 Chopped
B 16 Dec, 2018 Chopped
C 16 Dec, 2018 Chopped
D 16 Dec, 2018 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
6hsgA00 28 Feb, 2019 3.40.800.20 Assigned
6hsgB00 28 Feb, 2019 3.40.800.20 Assigned
6hsgC00 28 Feb, 2019 3.40.800.20 Assigned
6hsgD00 28 Feb, 2019 3.40.800.20 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
A5H660 A5H660_SCHMA Schistosoma mansoni Histone deacetylase 8
A5H660 A5H660_SCHMA Schistosoma mansoni Histone deacetylase 8
A5H660 A5H660_SCHMA Schistosoma mansoni Histone deacetylase 8
A5H660 A5H660_SCHMA Schistosoma mansoni Histone deacetylase 8