PDB Information

PDB6HKM
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery and Characterization of the Potent and Highly Selective (Piperidin-4-yl)pyrido[3,2- d]pyrimidine Based in Vitro Probe BAY-885 for the Kinase ERK5.
Nguyen, D., Lemos, C., Wortmann, L., Eis, K., Holton, S.J., Boemer, U., Moosmayer, D., Eberspaecher, U., Weiske, J., Lechner, C., Prechtl, S., Suelzle, D., Siegel, F., Prinz, F., Lesche, R., Nicke, B., Nowak-Reppel, K., Himmel, H., Mumberg, D., von Nussbaum, F., Nising, C.F., Bauser, M., Haegebarth, A.
J. Med. Chem.
HeaderTransferase
Released2018-09-07
Resolution2.470
CATH Insert Date03 Mar, 2019

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 03 Mar, 2019 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6hkmA01 04 Mar, 2019 3.30.200.20 Assigned
6hkmA02 04 Mar, 2019 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q13164 MK07_HUMAN Homo sapiens Mitogen-activated protein kinase 7