PDB 6gla
PDB Information
| PDB | 6GLA |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | Development, Optimization, and Structure-Activity Relationships of Covalent-Reversible JAK3 Inhibitors Based on a Tricyclic Imidazo[5,4- d]pyrrolo[2,3- b]pyridine Scaffold.
J. Med. Chem.
|
| Header | Transferase |
| Released | 2018-05-23 |
| Resolution | 1.920 |
| CATH Insert Date | 06 Jul, 2018 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 06 Jul, 2018 | Chopped |
| B | 06 Jul, 2018 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 6glaA01 | 19 Jul, 2018 | 3.30.200.20 | Assigned |
| 6glaA02 | 19 Jul, 2018 | 1.10.510.10 | Assigned |
| 6glaB01 | 19 Jul, 2018 | 3.30.200.20 | Assigned |
| 6glaB02 | 19 Jul, 2018 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P52333 | JAK3_HUMAN | Homo sapiens | Tyrosine-protein kinase JAK3 |
| P52333 | JAK3_HUMAN | Homo sapiens | Tyrosine-protein kinase JAK3 |
