PDB Information

PDB6G8N
MethodX-RAY DIFFRACTION
Host OrganismSaccharomyces cerevisiae
Gene SourceSaccharomyces cerevisiae (strain ATCC 204508 / S288c)
Primary Citation
Design, synthesis, and evaluation of cystargolide-based beta-lactones as potent proteasome inhibitors.
Niroula, D., Hallada, L.P., Le Chapelain, C., Ganegamage, S.K., Dotson, D., Rogelj, S., Groll, M., Tello-Aburto, R.
Eur J Med Chem
HeaderHydrolase
Released2018-04-09
Resolution3.000
CATH Insert Date16 Sep, 2018

PDB Images (57)

PDB Prints

PDB Chains (28)

Chain ID Date inserted into CATH CATH Status
a 16 Sep, 2018 Chopped
A 16 Sep, 2018 Chopped
b 16 Sep, 2018 Chopped
B 16 Sep, 2018 Chopped
C 16 Sep, 2018 Chopped
D 16 Sep, 2018 Chopped
E 16 Sep, 2018 Chopped
F 16 Sep, 2018 Chopped
G 16 Sep, 2018 Chopped
H 16 Sep, 2018 Chopped
I 16 Sep, 2018 Chopped
J 16 Sep, 2018 Chopped
K 16 Sep, 2018 Chopped
L 16 Sep, 2018 Chopped
M 16 Sep, 2018 Chopped
N 16 Sep, 2018 Chopped
O 16 Sep, 2018 Chopped
P 16 Sep, 2018 Chopped
Q 16 Sep, 2018 Chopped
R 16 Sep, 2018 Chopped
S 16 Sep, 2018 Chopped
T 16 Sep, 2018 Chopped
U 16 Sep, 2018 Chopped
V 16 Sep, 2018 Chopped
W 16 Sep, 2018 Chopped
X 16 Sep, 2018 Chopped
Y 16 Sep, 2018 Chopped
Z 16 Sep, 2018 Chopped

CATH Domains (28)

Domain ID Date inserted into CATH Superfamily CATH Status
6g8na00 17 Sep, 2018 3.60.20.10 Assigned
6g8nA00 17 Sep, 2018 3.60.20.10 Assigned
6g8nb00 17 Sep, 2018 3.60.20.10 Assigned
6g8nB00 17 Sep, 2018 3.60.20.10 Assigned
6g8nC00 17 Sep, 2018 3.60.20.10 Assigned
6g8nD00 17 Sep, 2018 3.60.20.10 Assigned
6g8nE00 17 Sep, 2018 3.60.20.10 Assigned
6g8nF00 17 Sep, 2018 3.60.20.10 Assigned
6g8nG00 17 Sep, 2018 3.60.20.10 Assigned
6g8nH00 17 Sep, 2018 3.60.20.10 Assigned
6g8nI00 17 Sep, 2018 3.60.20.10 Assigned
6g8nJ00 17 Sep, 2018 3.60.20.10 Assigned
6g8nK00 17 Sep, 2018 3.60.20.10 Assigned
6g8nL00 17 Sep, 2018 3.60.20.10 Assigned
6g8nM00 17 Sep, 2018 3.60.20.10 Assigned
6g8nN00 17 Sep, 2018 3.60.20.10 Assigned
6g8nO00 17 Sep, 2018 3.60.20.10 Assigned
6g8nP00 17 Sep, 2018 3.60.20.10 Assigned
6g8nQ00 17 Sep, 2018 3.60.20.10 Assigned
6g8nR00 17 Sep, 2018 3.60.20.10 Assigned
6g8nS00 17 Sep, 2018 3.60.20.10 Assigned
6g8nT00 17 Sep, 2018 3.60.20.10 Assigned
6g8nU00 17 Sep, 2018 3.60.20.10 Assigned
6g8nV00 17 Sep, 2018 3.60.20.10 Assigned
6g8nW00 17 Sep, 2018 3.60.20.10 Assigned
6g8nX00 17 Sep, 2018 3.60.20.10 Assigned
6g8nY00 17 Sep, 2018 3.60.20.10 Assigned
6g8nZ00 17 Sep, 2018 3.60.20.10 Assigned

UniProtKB Entries (28)

Accession Gene ID Taxon Description
P25043 PSB2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-2
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P25043 PSB2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-2
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4