Scaffold-Hopping Approach To Discover Potent, Selective, and Efficacious Inhibitors of NF-kappa B Inducing Kinase.
Blaquiere, N., Castanedo, G.M., Burch, J.D., Berezhkovskiy, L.M., Brightbill, H., Brown, S., Chan, C., Chiang, P.C., Crawford, J.J., Dong, T., Fan, P., Feng, J., Ghilardi, N., Godemann, R., Gogol, E., Grabbe, A., Hole, A.J., Hu, B., Hymowitz, S.G., Alaoui Ismaili, M.H., Le, H., Lee, P., Lee, W., Lin, X., Liu, N., McEwan, P.A., McKenzie, B., Silvestre, H.L., Suto, E., Sujatha-Bhaskar, S., Wu, G., Wu, L.C., Zhang, Y., Zhong, Z., Staben, S.T.
J. Med. Chem.