PDB Information

PDB6G4Y
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceMus musculus
Primary Citation
Scaffold-Hopping Approach To Discover Potent, Selective, and Efficacious Inhibitors of NF-kappa B Inducing Kinase.
Blaquiere, N., Castanedo, G.M., Burch, J.D., Berezhkovskiy, L.M., Brightbill, H., Brown, S., Chan, C., Chiang, P.C., Crawford, J.J., Dong, T., Fan, P., Feng, J., Ghilardi, N., Godemann, R., Gogol, E., Grabbe, A., Hole, A.J., Hu, B., Hymowitz, S.G., Alaoui Ismaili, M.H., Le, H., Lee, P., Lee, W., Lin, X., Liu, N., McEwan, P.A., McKenzie, B., Silvestre, H.L., Suto, E., Sujatha-Bhaskar, S., Wu, G., Wu, L.C., Zhang, Y., Zhong, Z., Staben, S.T.
J. Med. Chem.
HeaderTransferase
Released2018-03-28
Resolution2.650
CATH Insert Date06 Jul, 2018

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 06 Jul, 2018 Chopped
B 06 Jul, 2018 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
6g4yA01 19 Jul, 2018 3.30.200.20 Assigned
6g4yA02 19 Jul, 2018 1.10.510.10 Assigned
6g4yB01 19 Jul, 2018 3.30.200.20 Assigned
6g4yB02 19 Jul, 2018 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9WUL6 M3K14_MOUSE Mus musculus Mitogen-activated protein kinase kinase kinase 14
Q9WUL6 M3K14_MOUSE Mus musculus Mitogen-activated protein kinase kinase kinase 14