PDB Information

PDB6EW6
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli-Pichia pastoris shuttle vector pPpARG4
Gene SourceHomo sapiens
Primary Citation
Development of a Novel B-Cell Lymphoma 6 (BCL6) PROTAC To Provide Insight into Small Molecule Targeting of BCL6.
McCoull, W., Cheung, T., Anderson, E., Barton, P., Burgess, J., Byth, K., Cao, Q., Castaldi, M.P., Chen, H., Chiarparin, E., Carbajo, R.J., Code, E., Cowan, S., Davey, P.R., Ferguson, A.D., Fillery, S., Fuller, N.O., Gao, N., Hargreaves, D., Howard, M.R., Hu, J., Kawatkar, A., Kemmitt, P.D., Leo, E., Molina, D.M., O'Connell, N., Petteruti, P., Rasmusson, T., Raubo, P., Rawlins, P.B., Ricchiuto, P., Robb, G.R., Schenone, M., Waring, M.J., Zinda, M., Fawell, S., Wilson, D.M.
ACS Chem. Biol.
HeaderTransferase
Released2017-11-03
Resolution1.390
CATH Insert Date16 Dec, 2018

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Dec, 2018 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
6ew6A00 28 Feb, 2019 3.30.710.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P41182 BCL6_HUMAN Homo sapiens B-cell lymphoma 6 protein