PDB Information

PDB6EL7
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Discovery of a Novel Oral Glucocorticoid Receptor Modulator (AZD9567) with Improved Side Effect Profile.
Ripa, L., Edman, K., Dearman, M., Edenro, G., Hendrickx, R., Ullah, V., Chang, H.F., Lepisto, M., Chapman, D., Geschwindner, S., Wissler, L., Svanberg, P., Lawitz, K., Malmberg, J., Nikitidis, A., Olsson, R.I., Bird, J., Llinas, A., Hegelund-Myrback, T., Berger, M., Thorne, P., Harrison, R., Kohler, C., Drmota, T.
J. Med. Chem.
HeaderSignaling Protein
Released2017-09-28
Resolution2.180
CATH Insert Date03 Jun, 2018

PDB Images (4)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped
B 03 Jun, 2018 Rejected

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
6el7A00 29 Jun, 2018 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q15596 NCOA2_HUMAN Homo sapiens Nuclear receptor coactivator 2
P04150 GCR_HUMAN Homo sapiens Glucocorticoid receptor