PDB Information

PDB6E5G
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21
Gene SourceHomo sapiens
Primary Citation
Small-Molecule Covalent Modification of Conserved Cysteine Leads to Allosteric Inhibition of the TEAD⋅Yap Protein-Protein Interaction.
Bum-Erdene, K., Zhou, D., Gonzalez-Gutierrez, G., Ghozayel, M.K., Si, Y., Xu, D., Shannon, H.E., Bailey, B.J., Corson, T.W., Pollok, K.E., Wells, C.D., Meroueh, S.O.
Cell Chem Biol
HeaderTranscription/Inhibitor
Released2018-07-20
Resolution2.430
CATH Insert Date20 Jan, 2019

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 20 Jan, 2019 Chopped
B 20 Jan, 2019 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6e5gA00 21 Jan, 2019 2.70.50.80 Assigned
6e5gB00 21 Jan, 2019 2.70.50.80 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q15562 TEAD2_HUMAN Homo sapiens Transcriptional enhancer factor TEF-4
Q15562 TEAD2_HUMAN Homo sapiens Transcriptional enhancer factor TEF-4