PDB Information

PDB6E4A
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Discovery and lead identification of quinazoline-based BRD4 inhibitors.
Yang, S.M., Urban, D.J., Yoshioka, M., Strovel, J.W., Fletcher, S., Wang, A.Q., Xu, X., Shah, P., Hu, X., Hall, M.D., Jadhav, A., Maloney, D.J.
Bioorg. Med. Chem. Lett.
HeaderProtein Binding
Released2018-07-17
Resolution1.260
CATH Insert Date16 Sep, 2018

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 16 Sep, 2018 Chopped
B 16 Sep, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6e4aA01 17 Sep, 2018 1.20.920.10 Assigned
6e4aB01 17 Sep, 2018 1.20.920.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4