PDB 6e4a
PDB Information
| PDB | 6E4A |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21(DE3) |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery and lead identification of quinazoline-based BRD4 inhibitors.
Bioorg. Med. Chem. Lett.
|
| Header | Protein Binding |
| Released | 2018-07-17 |
| Resolution | 1.260 |
| CATH Insert Date | 16 Sep, 2018 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 16 Sep, 2018 | Chopped |
| B | 16 Sep, 2018 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 6e4aA01 | 17 Sep, 2018 | 1.20.920.10 | Assigned |
| 6e4aB01 | 17 Sep, 2018 | 1.20.920.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
| O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
