PDB Information

PDB6DB3
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Identification of Cyanamide-Based Janus Kinase 3 (JAK3) Covalent Inhibitors.
Casimiro-Garcia, A., Trujillo, J.I., Vajdos, F., Juba, B., Banker, M.E., Aulabaugh, A., Balbo, P., Bauman, J., Chrencik, J., Coe, J.W., Czerwinski, R., Dowty, M., Knafels, J.D., Kwon, S., Leung, L., Liang, S., Robinson, R.P., Telliez, J.B., Unwalla, R., Yang, X., Thorarensen, A.
J. Med. Chem.
HeaderTransferase/Inhibitor
Released2018-05-02
Resolution1.970
CATH Insert Date16 Dec, 2018

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Dec, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6db3A01 28 Feb, 2019 3.30.200.20 Assigned
6db3A02 28 Feb, 2019 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P52333 JAK3_HUMAN Homo sapiens Tyrosine-protein kinase JAK3