PDB Information

PDB6D8E
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery of a Highly Potent and Broadly Effective Epidermal Growth Factor Receptor and HER2 Exon 20 Insertion Mutant Inhibitor.
Jang, J., Son, J., Park, E., Kosaka, T., Saxon, J.A., De Clercq, D.J.H., Choi, H.G., Tanizaki, J., Eck, M.J., Janne, P.A., Gray, N.S.
Angew. Chem. Int. Ed. Engl.
HeaderTransferase/Transferase Inhibitor
Released2018-04-26
Resolution2.540
CATH Insert Date22 Jul, 2018

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 22 Jul, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6d8eA01 23 Jul, 2018 3.30.200.20 Assigned
6d8eA02 23 Jul, 2018 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P00533 EGFR_HUMAN Homo sapiens Epidermal growth factor receptor