PDB Information

PDB6D4Q
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceMycobacterium thermoresistibile (strain ATCC 19527 / DSM 44167 / CIP 105390 / JCM 6362 / NCTC 10409 / 316)
Primary Citation
Synthesis and Structure-Activity relationship of 1-(5-isoquinolinesulfonyl)piperazine analogues as inhibitors of Mycobacterium tuberculosis IMPDH.
Singh, V., Pacitto, A., Donini, S., Ferraris, D.M., Boros, S., Illyes, E., Szokol, B., Rizzi, M., Blundell, T.L., Ascher, D.B., Pato, J., Mizrahi, V.
Eur.J.Med.Chem.
HeaderOxidoreductase/Oxidoreductase Inhibitor
Released2018-04-18
Resolution1.710
CATH Insert Date05 May, 2019

PDB Images (2)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 May, 2019 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (1)

Accession Gene ID Taxon Description
G7CNL4 G7CNL4_MYCT3 Mycolicibacterium thermoresistibile ATCC 19527 Inosine-5'-monophosphate dehydrogenase