PDB 6ckr
PDB Information
PDB | 6CKR |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli K-12 |
Gene Source | Homo sapiens |
Primary Citation | Design, synthesis and biological evaluation of novel 4-phenylisoquinolinone BET bromodomain inhibitors.
Bioorg. Med. Chem. Lett.
|
Header | Gene Regulation/Inhibitor |
Released | 2018-02-28 |
Resolution | 1.620 |
CATH Insert Date | 03 Jun, 2018 |
PDB Images (5)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 03 Jun, 2018 | Chopped |
B | 03 Jun, 2018 | Chopped |
CATH Domains (2)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
6ckrA01 | 29 Jun, 2018 | 1.20.920.10 | Assigned |
6ckrB01 | 29 Jun, 2018 | 1.20.920.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |