PDB 6cg1
PDB Information
| PDB | 6CG1 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli K-12 |
| Gene Source | Homo sapiens |
| Primary Citation | Structure-based design and discovery of potent and selective KDM5 inhibitors.
Bioorg. Med. Chem. Lett.
|
| Header | Oxidoreductase/Inhibitor |
| Released | 2018-02-19 |
| Resolution | 2.160 |
| CATH Insert Date | 03 Jun, 2018 |
PDB Images (9)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 03 Jun, 2018 | Chopped |
| B | 03 Jun, 2018 | Chopped |
| C | 03 Jun, 2018 | Chopped |
| D | 03 Jun, 2018 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 6cg1A01 | 28 Jun, 2018 | 2.60.120.650 | Assigned |
| 6cg1B01 | 28 Jun, 2018 | 2.60.120.650 | Assigned |
| 6cg1C01 | 28 Jun, 2018 | 2.60.120.650 | Assigned |
| 6cg1D01 | 28 Jun, 2018 | 2.60.120.650 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O75164 | KDM4A_HUMAN | Homo sapiens | Lysine-specific demethylase 4A |
| O75164 | KDM4A_HUMAN | Homo sapiens | Lysine-specific demethylase 4A |
| O75164 | KDM4A_HUMAN | Homo sapiens | Lysine-specific demethylase 4A |
| O75164 | KDM4A_HUMAN | Homo sapiens | Lysine-specific demethylase 4A |
