PDB Information

PDB6BVL
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of Aminopiperidine Indoles That Activate the Guanine Nucleotide Exchange Factor SOS1 and Modulate RAS Signaling.
Abbott, J.R., Hodges, T.R., Daniels, R.N., Patel, P.A., Kennedy, J.P., Howes, J.E., Akan, D.T., Burns, M.C., Sai, J., Sobolik, T., Beesetty, Y., Lee, T., Rossanese, O.W., Phan, J., Waterson, A.G., Fesik, S.W.
J. Med. Chem.
HeaderSignaling Protein
Released2017-12-13
Resolution1.750
CATH Insert Date16 Dec, 2018

PDB Images (8)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
A 16 Dec, 2018 Chopped
B 16 Dec, 2018 Chopped
C 16 Dec, 2018 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
6bvlA00 28 Feb, 2019 3.40.50.300 Assigned
6bvlB01 28 Feb, 2019 1.20.870.10 Assigned
6bvlB02 28 Feb, 2019 1.10.840.10 Assigned
6bvlC00 28 Feb, 2019 3.40.50.300 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
Q07889 SOS1_HUMAN Homo sapiens Son of sevenless homolog 1
P01112 RASH_HUMAN Homo sapiens GTPase HRas
P01112 RASH_HUMAN Homo sapiens GTPase HRas