PDB Information

PDB6B1X
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceKlebsiella pneumoniae
Primary Citation
Strategic Approaches to Overcome Resistance against Gram-Negative Pathogens Using beta-Lactamase Inhibitors and beta-Lactam Enhancers: Activity of Three Novel Diazabicyclooctanes WCK 5153, Zidebactam (WCK 5107), and WCK 4234.
Papp-Wallace, K.M., Nguyen, N.Q., Jacobs, M.R., Bethel, C.R., Barnes, M.D., Kumar, V., Bajaksouzian, S., Rudin, S.D., Rather, P.N., Bhavsar, S., Ravikumar, T., Deshpande, P.K., Patil, V., Yeole, R., Bhagwat, S.S., Patel, M.V., van den Akker, F., Bonomo, R.A.
J. Med. Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2017-09-19
Resolution1.450
CATH Insert Date05 Aug, 2018

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Aug, 2018 Chopped
B 05 Aug, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6b1xA00 06 Aug, 2018 3.40.710.10 Assigned
6b1xB00 06 Aug, 2018 3.40.710.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9F663 BLKPC_KLEPN Klebsiella pneumoniae Carbapenem-hydrolyzing beta-lactamase KPC
Q9F663 BLKPC_KLEPN Klebsiella pneumoniae Carbapenem-hydrolyzing beta-lactamase KPC