PDB Information

PDB6ACR
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Bis-Heteroaryl Pyrazoles: Identification of Orally Bioavailable Inhibitors of Activin Receptor-Like Kinase-2 (R206H).
Sekimata, K., Sato, T., Sakai, N., Watanabe, H., Mishima-Tsumagari, C., Taguri, T., Matsumoto, T., Fujii, Y., Handa, N., Honma, T., Tanaka, A., Shirouzu, M., Yokoyama, S., Miyazono, K., Hashizume, Y., Koyama, H.
Chem. Pharm. Bull.
HeaderSignaling Protein
Released2018-07-27
Resolution2.010
CATH Insert Date24 Mar, 2019

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 24 Mar, 2019 Chopped
B 24 Mar, 2019 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
6acrA01 25 Mar, 2019 3.30.200.20 Assigned
6acrA02 25 Mar, 2019 1.10.510.10 Assigned
6acrB01 25 Mar, 2019 3.30.200.20 Assigned
6acrB02 25 Mar, 2019 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q04771 ACVR1_HUMAN Homo sapiens Activin receptor type-1
Q04771 ACVR1_HUMAN Homo sapiens Activin receptor type-1