PDB 6a3n
PDB Information
| PDB | 6A3N |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21 |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of Potent, Selective, and Orally Bioavailable Inhibitors against Phosphodiesterase-9, a Novel Target for the Treatment of Vascular Dementia.
J. Med. Chem.
|
| Header | Hydrolase |
| Released | 2018-06-15 |
| Resolution | 2.600 |
| CATH Insert Date | 14 Apr, 2019 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 14 Apr, 2019 | Chopped |
| B | 14 Apr, 2019 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 6a3nA00 | 15 Apr, 2019 | 1.10.1300.10 | Assigned |
| 6a3nB00 | 15 Apr, 2019 | 1.10.1300.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O76083 | PDE9A_HUMAN | Homo sapiens | High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A |
| O76083 | PDE9A_HUMAN | Homo sapiens | High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A |
