PDB 5zz4
PDB Information
| PDB | 5ZZ4 |
| Method | X-RAY DIFFRACTION |
| Host Organism | unidentified baculovirus |
| Gene Source | Homo sapiens |
| Primary Citation | Design and Synthesis of Novel Amino-triazine Analogues as Selective Bruton's Tyrosine Kinase Inhibitors for Treatment of Rheumatoid Arthritis.
J. Med. Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2018-05-30 |
| Resolution | 2.900 |
| CATH Insert Date | 30 Sep, 2018 |
PDB Images (19)
PDB Prints
PDB Chains (6)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 30 Sep, 2018 | Chopped |
| B | 30 Sep, 2018 | Chopped |
| C | 30 Sep, 2018 | Chopped |
| D | 30 Sep, 2018 | Chopped |
| E | 30 Sep, 2018 | Chopped |
| F | 30 Sep, 2018 | Chopped |
CATH Domains (12)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5zz4A01 | 01 Oct, 2018 | 3.30.200.20 | Assigned |
| 5zz4A02 | 01 Oct, 2018 | 1.10.510.10 | Assigned |
| 5zz4B01 | 01 Oct, 2018 | 3.30.200.20 | Assigned |
| 5zz4B02 | 01 Oct, 2018 | 1.10.510.10 | Assigned |
| 5zz4C01 | 01 Oct, 2018 | 3.30.200.20 | Assigned |
| 5zz4C02 | 01 Oct, 2018 | 1.10.510.10 | Assigned |
| 5zz4D01 | 01 Oct, 2018 | 3.30.200.20 | Assigned |
| 5zz4D02 | 01 Oct, 2018 | 1.10.510.10 | Assigned |
| 5zz4E01 | 01 Oct, 2018 | 3.30.200.20 | Assigned |
| 5zz4E02 | 01 Oct, 2018 | 1.10.510.10 | Assigned |
| 5zz4F01 | 01 Oct, 2018 | 3.30.200.20 | Assigned |
| 5zz4F02 | 01 Oct, 2018 | 1.10.510.10 | Assigned |
UniProtKB Entries (6)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q06187 | BTK_HUMAN | Homo sapiens | Tyrosine-protein kinase BTK |
| Q06187 | BTK_HUMAN | Homo sapiens | Tyrosine-protein kinase BTK |
| Q06187 | BTK_HUMAN | Homo sapiens | Tyrosine-protein kinase BTK |
| Q06187 | BTK_HUMAN | Homo sapiens | Tyrosine-protein kinase BTK |
| Q06187 | BTK_HUMAN | Homo sapiens | Tyrosine-protein kinase BTK |
| Q06187 | BTK_HUMAN | Homo sapiens | Tyrosine-protein kinase BTK |
