PDB Information

PDB5Z5U
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Development and evaluation of a novel series of Nitroxoline-derived BET inhibitors with antitumor activity in renal cell carcinoma.
Chen, W., Zhang, H., Chen, Z., Jiang, H., Liao, L., Fan, S., Xing, J., Xie, Y., Chen, S., Ding, H., Chen, K., Jiang, H., Luo, C., Zheng, M., Yao, Z., Huang, Y., Zhang, Y.
Oncogenesis
HeaderTranscription/Inhibitor
Released2018-01-20
Resolution1.630
CATH Insert Date27 Jan, 2019

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 27 Jan, 2019 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5z5uA01 28 Jan, 2019 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4