PDB Information

PDB5Z5S
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of DS-6930, a potent selective PPAR gamma modulator. Part I: Lead identification.
Shinozuka, T., Tsukada, T., Fujii, K., Tokumaru, E., Shimada, K., Onishi, Y., Matsui, Y., Wakimoto, S., Kuroha, M., Ogata, T., Araki, K., Ohsumi, J., Sawamura, R., Watanabe, N., Yamamoto, H., Fujimoto, K., Tani, Y., Mori, M., Tanaka, J.
Bioorg. Med. Chem.
HeaderTranscription
Released2018-01-19
Resolution1.800
CATH Insert Date16 Dec, 2018

PDB Images (4)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 16 Dec, 2018 Chopped
C 16 Dec, 2018 Rejected

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5z5sA00 28 Feb, 2019 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9UBK2 PRGC1_HUMAN Homo sapiens Peroxisome proliferator-activated receptor gamma coactivator 1-alpha
P37231 PPARG_HUMAN Homo sapiens Peroxisome proliferator-activated receptor gamma