PDB Information

PDB5Z1R
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21
Gene SourceHomo sapiens
Primary Citation
Y08060: A Selective BET Inhibitor for Treatment of Prostate Cancer.
Xiang, Q., Zhang, Y., Li, J., Xue, X., Wang, C., Song, M., Zhang, C., Wang, R., Li, C., Wu, C., Zhou, Y., Yang, X., Li, G., Ding, K., Xu, Y.
Acs Med.Chem.Lett.
HeaderTranscription
Released2017-12-28
Resolution1.620
CATH Insert Date06 Jan, 2019

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 06 Jan, 2019 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5z1rA01 07 Jan, 2019 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4