PDB Information

PDB5YU9
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Ibrutinib targets mutant-EGFR kinase with a distinct binding conformation.
Wang, A., Yan, X.E., Wu, H., Wang, W., Hu, C., Chen, C., Zhao, Z., Zhao, P., Li, X., Wang, L., Wang, B., Ye, Z., Wang, J., Wang, C., Zhang, W., Gray, N.S., Weisberg, E.L., Chen, L., Liu, J., Yun, C.H., Liu, Q.
Oncotarget
HeaderOncoprotein
Released2017-11-21
Resolution1.950
CATH Insert Date07 Jan, 2018

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 07 Jan, 2018 Chopped
B 07 Jan, 2018 Chopped
C 07 Jan, 2018 Chopped
D 07 Jan, 2018 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
5yu9A01 11 Jan, 2018 3.30.200.20 Assigned
5yu9A02 11 Jan, 2018 1.10.510.10 Assigned
5yu9B01 11 Jan, 2018 3.30.200.20 Assigned
5yu9B02 11 Jan, 2018 1.10.510.10 Assigned
5yu9C01 11 Jan, 2018 3.30.200.20 Assigned
5yu9C02 11 Jan, 2018 1.10.510.10 Assigned
5yu9D01 11 Jan, 2018 3.30.200.20 Assigned
5yu9D02 11 Jan, 2018 1.10.510.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P00533 EGFR_HUMAN Homo sapiens Epidermal growth factor receptor
P00533 EGFR_HUMAN Homo sapiens Epidermal growth factor receptor
P00533 EGFR_HUMAN Homo sapiens Epidermal growth factor receptor
P00533 EGFR_HUMAN Homo sapiens Epidermal growth factor receptor