PDB Information

PDB5Y1Y
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of novel BET inhibitors by drug repurposing of nitroxoline and its analogues.
Jiang, H., Xing, J., Wang, C., Zhang, H., Yue, L., Wan, X., Chen, W., Ding, H., Xie, Y., Tao, H., Chen, Z., Jiang, H., Chen, K., Chen, S., Zheng, M., Zhang, Y., Luo, C.
Org. Biomol. Chem.
HeaderTranscription
Released2017-07-21
Resolution1.910
CATH Insert Date17 Dec, 2017

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 17 Dec, 2017 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5y1yA01 23 Dec, 2017 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4