PDB Information

PDB5X5O
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Structure Based Design of N-(3-((1H-Pyrazolo[3,4-b]pyridin-5-yl)ethynyl)benzenesulfonamides as Selective Leucine-Zipper and Sterile-alpha Motif Kinase (ZAK) Inhibitors.
Chang, Y., Lu, X., Shibu, M.A., Dai, Y.B., Luo, J., Zhang, Y., Li, Y., Zhao, P., Zhang, Z., Xu, Y., Tu, Z.C., Zhang, Q.W., Yun, C.H., Huang, C.Y., Ding, K.
J. Med. Chem.
HeaderTransferase
Released2017-02-17
Resolution1.870
CATH Insert Date07 Jan, 2018

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 07 Jan, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5x5oA01 11 Jan, 2018 3.30.200.20 Assigned
5x5oA02 11 Jan, 2018 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9NYL2 M3K20_HUMAN Homo sapiens Mitogen-activated protein kinase kinase kinase 20