PDB Information

PDB5WMT
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceCanis lupus familiaris
Primary Citation
Structure Based Design of a Grp94-Selective Inhibitor: Exploiting a Key Residue in Grp94 To Optimize Paralog-Selective Binding.
Que, N.L.S., Crowley, V.M., Duerfeldt, A.S., Zhao, J., Kent, C.N., Blagg, B.S.J., Gewirth, D.T.
J. Med. Chem.
HeaderChaperone/Inhibitor
Released2017-07-31
Resolution2.750
CATH Insert Date03 Jun, 2018

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped
B 03 Jun, 2018 Chopped
C 03 Jun, 2018 Chopped
D 03 Jun, 2018 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5wmtA00 28 Jun, 2018 3.30.565.10 Assigned
5wmtB00 28 Jun, 2018 3.30.565.10 Assigned
5wmtC00 28 Jun, 2018 3.30.565.10 Assigned
5wmtD00 28 Jun, 2018 3.30.565.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P41148 ENPL_CANLF Canis lupus familiaris Endoplasmin
P41148 ENPL_CANLF Canis lupus familiaris Endoplasmin
P41148 ENPL_CANLF Canis lupus familiaris Endoplasmin
P41148 ENPL_CANLF Canis lupus familiaris Endoplasmin