PDB Information

PDB5WJ6
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Characterization of the interactions of potent allosteric inhibitors with glutaminase C, a key enzyme in cancer cell glutamine metabolism.
Huang, Q., Stalnecker, C., Zhang, C., McDermott, L.A., Iyer, P., O'Neill, J., Reimer, S., Cerione, R.A., Katt, W.P.
J. Biol. Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2017-07-21
Resolution2.450
CATH Insert Date03 Jun, 2018

PDB Images (5)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Holding pen
B 03 Jun, 2018 Holding pen
C 03 Jun, 2018 Holding pen
D 03 Jun, 2018 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (4)

Accession Gene ID Taxon Description
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial