PDB Information

PDB5WG8
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
The Antitumor Drug LB-100 Is a Catalytic Inhibitor of Protein Phosphatase 2A (PPP2CA) and 5 (PPP5C) Coordinating with the Active-Site Catalytic Metals in PPP5C.
D'Arcy, B.M., Swingle, M.R., Papke, C.M., Abney, K.A., Bouska, E.S., Prakash, A., Honkanen, R.E.
Mol. Cancer Ther.
HeaderHydrolase/Hydrolase Inhibitor
Released2017-07-13
Resolution1.650
CATH Insert Date22 Jul, 2018

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 22 Jul, 2018 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5wg8A00 23 Jul, 2018 3.60.21.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P53041 PPP5_HUMAN Homo sapiens Serine/threonine-protein phosphatase 5