PDB Information

PDB5W0I
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceMus musculus
Primary Citation
GNE-781, A Highly Advanced Potent and Selective Bromodomain Inhibitor of Cyclic Adenosine Monophosphate Response Element Binding Protein, Binding Protein (CBP).
Romero, F.A., Murray, J., Lai, K.W., Tsui, V., Albrecht, B.K., An, L., Beresini, M.H., de Leon Boenig, G., Bronner, S.M., Chan, E.W., Chen, K.X., Chen, Z., Choo, E.F., Clagg, K., Clark, K., Crawford, T.D., Cyr, P., de Almeida Nagata, D., Gascoigne, K.E., Grogan, J.L., Hatzivassiliou, G., Huang, W., Hunsaker, T.L., Kaufman, S., Koenig, S.G., Li, R., Li, Y., Liang, X., Liao, J., Liu, W., Ly, J., Maher, J., Masui, C., Merchant, M., Ran, Y., Taylor, A.M., Wai, J., Wang, F., Wei, X., Yu, D., Zhu, B.Y., Zhu, X., Magnuson, S.
J. Med. Chem.
HeaderTransferase/Inhibitor
Released2017-05-30
Resolution1.430
CATH Insert Date03 Jun, 2018

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5w0iA00 28 Jun, 2018 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P45481 CBP_MOUSE Mus musculus CREB-binding protein