PDB Information

PDB5VZS
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
GNE-781, A Highly Advanced Potent and Selective Bromodomain Inhibitor of CBP/P300
Murray, J.M.
To be published
HeaderTranscription Regulator/Inhibitor
Released2017-05-29
Resolution1.710
CATH Insert Date06 Jul, 2018

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 06 Jul, 2018 Chopped
B 06 Jul, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5vzsA01 19 Jul, 2018 1.20.920.10 Assigned
5vzsB01 19 Jul, 2018 1.20.920.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4