PDB Information

PDB5V8R
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceClostridium botulinum
Primary Citation
Small molecule metalloprotease inhibitor with in vitro, ex vivo and in vivo efficacy against botulinum neurotoxin serotype A.
Jacobson, A.R., Adler, M., Silvaggi, N.R., Allen, K.N., Smith, G.M., Fredenburg, R.A., Stein, R.L., Park, J.B., Feng, X., Shoemaker, C.B., Deshpande, S.S., Goodnough, M.C., Malizio, C.J., Johnson, E.A., Pellett, S., Tepp, W.H., Tzipori, S.
Toxicon
HeaderHydrolase/Hydrolase Inhibitor
Released2017-03-22
Resolution1.900
CATH Insert Date14 Nov, 2017

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped
B 14 Nov, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5v8rA01 10 Dec, 2017 3.90.1240.10 Assigned
5v8rB01 10 Dec, 2017 3.90.1240.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P0DPI1 BXA1_CLOBH Clostridium botulinum A str. Hall Botulinum neurotoxin type A
P0DPI1 BXA1_CLOBH Clostridium botulinum A str. Hall Botulinum neurotoxin type A