PDB 5v24
PDB Information
| PDB | 5V24 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Structure-based drug design of novel ASK1 inhibitors using an integrated lead optimization strategy.
Bioorg. Med. Chem. Lett.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2017-03-02 |
| Resolution | 2.500 |
| CATH Insert Date | 07 May, 2017 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 May, 2017 | Chopped |
| B | 08 May, 2017 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5v24A01 | 26 May, 2017 | 3.30.200.20 | Assigned |
| 5v24A02 | 26 May, 2017 | 1.10.510.10 | Assigned |
| 5v24B01 | 26 May, 2017 | 3.30.200.20 | Assigned |
| 5v24B02 | 26 May, 2017 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q99683 | M3K5_HUMAN | Homo sapiens | Mitogen-activated protein kinase kinase kinase 5 |
| Q99683 | M3K5_HUMAN | Homo sapiens | Mitogen-activated protein kinase kinase kinase 5 |
