PDB Information

PDB5V1B
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
1,2,4-Triazolo-[1,5-a]pyridine HIF Prolylhydroxylase Domain-1 (PHD-1) Inhibitors With a Novel Monodentate Binding Interaction.
Ahmed, S., Ayscough, A., Barker, G.R., Canning, H.E., Davenport, R., Downham, R., Harrison, D., Jenkins, K., Kinsella, N., Livermore, D.G., Wright, S., Ivetac, A.D., Skene, R., Wilkens, S.J., Webster, N.A., Hendrick, A.G.
J. Med. Chem.
HeaderOxidoreductase/Inhibitor
Released2017-03-01
Resolution2.490
CATH Insert Date14 Nov, 2017

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5v1bA00 10 Dec, 2017 2.60.120.620 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q96KS0 EGLN2_HUMAN Homo sapiens Egl nine homolog 2