PDB 5uvc
PDB Information
| PDB | 5UVC |
| Method | X-RAY DIFFRACTION |
| Host Organism | Baculovirus expression vector pFastBac1-HM |
| Gene Source | Homo sapiens |
| Primary Citation | Design, Synthesis, and Evaluation of the Highly Selective and Potent G-Protein-Coupled Receptor Kinase 2 (GRK2) Inhibitor for the Potential Treatment of Heart Failure.
J. Med. Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2017-02-20 |
| Resolution | 2.650 |
| CATH Insert Date | 14 Nov, 2017 |
PDB Images (2)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 14 Nov, 2017 | Holding pen |
CATH Domains (0)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P25098 | ARBK1_HUMAN | Homo sapiens | Beta-adrenergic receptor kinase 1 |
